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A-17
CAS No. 505057-98-7
A-17( Hsp90α inhibitor A17 )
Catalog No. M14721 CAS No. 505057-98-7
A potent Hsp90α/p23 interaction inhibitor with IC50 of 0.15 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameA-17
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NoteResearch use only, not for human use.
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Brief DescriptionA potent Hsp90α/p23 interaction inhibitor with IC50 of 0.15 uM.
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DescriptionA potent Hsp90α/p23 interaction inhibitor with IC50 of 0.15 uM, more effective than CP-9 in degrading pAkt/total Akt and Raf-1; inhibits Hsp90(α/β)/p23 interactions and degrading Hsp90 client proteins in cell culture, but not in live mice.
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In Vitro——
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In Vivo——
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SynonymsHsp90α inhibitor A17
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetHSP
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RecptorHSP
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Research Area——
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Indication——
Chemical Information
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CAS Number505057-98-7
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Formula Weight384.333
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Molecular FormulaC15H11F3N4O3S
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name2-((4-(furan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl)thio)-N-(5-methylisoxazol-3-yl)acetamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Chan CT, et al. Proc Natl Acad Sci U S A. 2012 Sep 11;109(37):E2476-85.
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