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(R)-Baclofen

CAS No. 69308-37-8

(R)-Baclofen( STX-209 )

Catalog No. M15651 CAS No. 69308-37-8

A derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist; also blocks α2δ subunit-containing voltage-dependent calcium channel (VDCC) with Ki of 156 uM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
5MG	30	In Stock
10MG	49	In Stock
25MG	101	In Stock
50MG	170	In Stock
100MG	265	In Stock
200MG	399	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

(R)-Baclofen
Note

Research use only, not for human use.
Brief Description

A derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist; also blocks α2δ subunit-containing voltage-dependent calcium channel (VDCC) with Ki of 156 uM.
Description

A derivative of the neurotransmitter GABA that acts as a GABAB receptor agonist; also blocks α2δ subunit-containing voltage-dependent calcium channel (VDCC) with Ki of 156 uM; A neurotransmitter inhibitor by blocking the release of excitatory transmitters; serves as a central nervous system depressant and skeletal muscle relaxant.Other Indication Approved.
In Vitro

——
In Vivo

——
Synonyms

STX-209
Pathway

Membrane Transporter/Ion Channel
Target

GAT
Recptor

GABAR
Research Area

Other Indications
Indication

Other Disease

Chemical Information

CAS Number

69308-37-8
Formula Weight

213.6608
Molecular Formula

C10H12ClNO2
Purity

>98% (HPLC)
Solubility

H2O: 5 mg/mL (Need ultrasonic)
SMILES

O=C(O)C[C@H](C1=CC=C(Cl)C=C1)CN
Chemical Name

Benzenepropanoic acid, β-(aminomethyl)-4-chloro-, (βR)-

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Zvejniece L, et al. Pharmacol Biochem Behav. 2015 Oct;137:23-9. 2. Carter LP, et al. Pharmacol Ther. 2009 Jan;121(1):100-14.

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