Cart
sales@molnova.com
Zuclopenthixol
CAS No. 53772-83-1
Zuclopenthixol ( alpha-Clopenthixol; Clopenthixol; Zuclopenthixol )
Catalog No. M18758 CAS No. 53772-83-1
Zuclopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 25MG | 27 | In Stock |
|
| 50MG | 35 | In Stock |
|
| 100MG | 50 | In Stock |
|
| 200MG | 72 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameZuclopenthixol
-
NoteResearch use only, not for human use.
-
Brief DescriptionZuclopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
-
DescriptionZuclopenthixol, also known as Cisordinol, Clopixol, Acuphase, zuclopentixol, is a typical antipsychotic drug of the thioxanthene class. It was introduced in 1962 by Lundbeck. Zuclopenthixol is the cis-isomer of clopenthixol. Zuclopenthixol is not approved for use in the United States. Zuclopenthixol has high affinity for both dopamine D1 and D2 receptors, for α1-adrenoceptors and 5-HT2 receptors but no affinity for cholinergic muscarine receptors. It has weak histamine (H1) receptor affinity and no α2-adrenoceptor blocking activity.
-
Synonymsalpha-Clopenthixol; Clopenthixol; Zuclopenthixol
-
PathwayOthers
-
TargetOther Targets
-
RecptorD1; D2
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number53772-83-1
-
Formula Weight400.96
-
Molecular FormulaC22H25ClN2OS
-
Purity98%
-
SolubilityDMSO : ≥ 150 mg/mL; 374.10 mM
-
SMILESC1CN(CCN1CC/C=C\1/c2ccccc2Sc2c1cc(cc2)Cl)CCO
-
Chemical Name2-[4-[(3Z)-3-(2-chlorothioxanthen-9-ylidene)propyl]piperazin-1-yl]ethanol
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Khalifa AE: Zuclopenthixol facilitates memory retrieval in rats: possible involvement of noradrenergic and serotonergic mechanisms. Pharmacol Biochem Behav. 2003 Jul;75(4):755-62.
molnova catalog
related products
-
CL 218872
CL 218872 is a benzodiazepine agonist displaying selectivity for α1 subunit-containing GABAA receptors (Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 nM for α1, α2, α3, α4, α5 and α6-subunit containing receptors respectively).
-
(E)-N-Caffeoylputres...
N-Caffeoylputrescine has antioxidant activity.
-
Prasugrel Hydrochlor...
Prasugrel hydrochloride is a piperazine derivative and pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.
