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YYA-021
CAS No. 144217-65-2
YYA-021( YYA 021 | YYA021 )
Catalog No. M11874 CAS No. 144217-65-2
A small-molecule CD4 mimic that acts as a highly potent HIV entry inhibitor with IC50 of 9 uM against YTA48P virus with no significant cytotoxicity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 33 | In Stock |
|
| 5MG | 53 | In Stock |
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| 10MG | 65 | In Stock |
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| 25MG | 140 | In Stock |
|
| 50MG | 194 | In Stock |
|
| 100MG | 250 | In Stock |
|
| 500MG | 614 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameYYA-021
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NoteResearch use only, not for human use.
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Brief DescriptionA small-molecule CD4 mimic that acts as a highly potent HIV entry inhibitor with IC50 of 9 uM against YTA48P virus with no significant cytotoxicity.
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DescriptionA small-molecule CD4 mimic that acts as a highly potent HIV entry inhibitor with IC50 of 9 uM against YTA48P virus with no significant cytotoxicity; shows wide tissue distribution and relatively high distribution volumes, and has promise for intravenous administration.
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In Vitro——
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In Vivo——
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SynonymsYYA 021 | YYA021
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PathwayMicrobiology/Virology
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TargetHIV
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RecptorGp120
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Research AreaInfection
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Indication——
Chemical Information
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CAS Number144217-65-2
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Formula Weight317.4259
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Molecular FormulaC18H27N3O2
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESO=C(NC1CC(C)(C)NC(C)(C)C1)C(NC2=CC=C(C)C=C2)=O
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Chemical NameEthanediamide, N1-(4-methylphenyl)-N2-(2,2,6,6-tetramethyl-4-piperidinyl)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Hashimoto C, et al. Bioorg Med Chem. 2013 Dec 15;21(24):7884-9.
2. Otsuki H, et al. J Gen Virol. 2013 Dec;94(Pt 12):2710-6.
3. Narumi T, et al. Bioorg Med Chem. 2013 May 1;21(9):2518-26.
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