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Vazegepant

CAS No. 1337918-83-8

Vazegepant( —— )

Catalog No. M35066 CAS No. 1337918-83-8

Vazegepant (Zavegepant) is an orally available and selective antagonist of the calcitonin gene-related peptide CGRP receptor for pain relief and may be used in the study of migraine.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 161 Get Quote
5MG 227 Get Quote
10MG 337 Get Quote
25MG 593 Get Quote
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Biological Information

  • Product Name
    Vazegepant
  • Note
    Research use only, not for human use.
  • Brief Description
    Vazegepant (Zavegepant) is an orally available and selective antagonist of the calcitonin gene-related peptide CGRP receptor for pain relief and may be used in the study of migraine.
  • Description
    Vazegepant (Zavegepant) is an orally active calcitonin gene-related peptideCGRP receptor antagonist with potential for acute research in migraine. CGRP is an important trigger in migraine pathophysiology.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    CGRP Receptor
  • Recptor
    CGRP Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1337918-83-8
  • Formula Weight
    638.8
  • Molecular Formula
    C36H46N8O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C1C(=CC=2C(N1)=CC=CC2)C3CCN(C(N[C@H](CC=4C=C5C(=C(C)C4)NN=C5)C(=O)N6CCN(CC6)C7CCN(C)CC7)=O)CC3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Leonard KA, et al. Discovery of a Gut-Restricted JAK Inhibitor for the Treatment of Inflammatory Bowel Disease. J Med Chem. 2020 Mar 26;63(6):2915-2929.?
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