VX-150
CAS No. 1793080-72-4
VX-150 ( —— )
Catalog No. M28830 CAS No. 1793080-72-4
VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 222 | Get Quote |
|
10MG | 356 | Get Quote |
|
25MG | 599 | Get Quote |
|
50MG | 852 | Get Quote |
|
100MG | 1152 | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameVX-150
-
NoteResearch use only, not for human use.
-
Brief DescriptionVX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).
-
DescriptionVX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).
-
Synonyms——
-
PathwayMembrane Transporter/Ion Channel
-
TargetSodium Channel
-
RecptorFatty Acid Synthase (FASN)
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number1793080-72-4
-
Formula Weight516.3
-
Molecular FormulaC21H17F4N2O7P
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCc(cc(cc1)F)c1Oc(cc(C(F)(F)F)cc1)c1C(NC(C=CN1COP(O)(O)=O)=CC1=O)=O
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Rae C, et al. Inhibition of Fatty Acid Synthase Sensitizes Prostate Cancer Cells to Radiotherapy. Radiat Res. 2015 Nov;184(5):482-93.
molnova catalog
related products
-
Veratridine
Veratridine is a benzoate-cevane found in veratrumand Schoenocaulon. It activates sodium channels to stay open longer than normal.
-
Tetracaine hydrochlo...
Tetracaine hydrochloride (Pontocaine) is a hydrochloride salt form of tetracaine which is a potent local anaesthetic and a channel function allosteric inhibitor.
-
APETx2
Acid-sensing ion channel 3 (ASIC3) channel blocker (IC50 values are 63 and 175 nM for homomeric rat and human ASIC3 channels). Also inhibits NaV1.8 and NaV1.2 channels (IC50 values are 55 and 114 nM respectively). Demonstrates analgesic properties against acid-induced and inflammatory pain.