VU 0255035( VU 255035 )

Catalog No. M27733 CAS No. 1135243-19-4

VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
5MG	65	In Stock
10MG	110	In Stock
25MG	233	In Stock
50MG	347	In Stock
100MG	511	In Stock
500MG	1062	In Stock
1G	Get Quote	In Stock

Get Quotation Bulk Inquiry Add to Cart

Biological Information

Product Name

VU 0255035
Note

Research use only, not for human use.
Brief Description

VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.
Description

VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM. It reduces pilocarpine-induced seizures in mice. It is used to examine the role of the M1 receptor in diverse situations.
In Vitro

——
In Vivo

——
Synonyms

VU 255035
Pathway

Cell Cycle/DNA Damage
Target

AChR
Recptor

——
Research Area

——
Indication

——

Chemical Information

CAS Number

1135243-19-4
Formula Weight

432.52
Molecular Formula

C18H20N6O3S2
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 62.5 mg/mL (144.50 mM)
SMILES

O=C(CCNS(=O)(=O)c1cccc2nsnc12)N1CCN(CC1)c1ccncc1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Yang YJ, et al. Effective Killing of Cancer Cells Through ROS-Mediated Mechanisms by AMRI-59 Targeting Peroxiredoxin I. Antioxid Redox Signal. 2016 Mar 10;24(8):453-69.

Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog

Product			Quantity Required*
Name *			E-mail Address *
Organization *			Phone Number
Remarks