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VAS2870
CAS No. 722456-31-7
VAS2870( VAS 2870 )
Catalog No. M17580 CAS No. 722456-31-7
VAS2870 is a NADPH oxidase (NOX) inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 47 | In Stock |
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| 10MG | 88 | In Stock |
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| 25MG | 170 | In Stock |
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| 50MG | 311 | In Stock |
|
| 100MG | 464 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameVAS2870
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NoteResearch use only, not for human use.
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Brief DescriptionVAS2870 is a NADPH oxidase (NOX) inhibitor.
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DescriptionVAS 2870 is a NADPH oxidase (Nox) inhibitor that enhances TGF-β-induced apoptosis of liver tumor cells.
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In Vitro——
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In Vivo——
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SynonymsVAS 2870
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PathwayPI3K/Akt/mTOR signaling
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TargetGSK-3
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RecptorNADPH oxidase (NOX)
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Research AreaCardiovascular Disease
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Indication——
Chemical Information
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CAS Number722456-31-7
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Formula Weight360.4
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Molecular FormulaC18H12N6OS
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Purity>98% (HPLC)
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SolubilityDMSO : 83.3 mg/mL. 231.14 mM;
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SMILESC12=C(SC3=NC4=C(C=CC=C4)O3)N=CN=C1N(CC5=CC=CC=C5)N=N2
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Chemical Name7-(2-Benzoxazolylthio)-3-(phenylmethyl)-3H-1,2,3-triazolo[4,5-d]pyrimidine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.ten Freyhaus H, et al. Novel Nox inhibitor VAS2870 attenuates PDGF-dependent smooth muscle cell chemotaxis, but not proliferation. Cardiovasc Res. 2006 Jul 15;71(2):331-41.
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