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UniPR505
CAS No. 2938227-14-4
UniPR505( —— )
Catalog No. M36518 CAS No. 2938227-14-4
UniPR505 is a potent EphA2 antagonist (IC50: 0.95 μM), a novel 3α-carbamoyloxy derivative with antiangiogenic properties.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 787 | Get Quote |
|
| 5MG | 1112 | Get Quote |
|
| 25MG | 1766 | Get Quote |
|
| 50MG | 2190 | Get Quote |
|
| 100MG | 2790 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameUniPR505
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NoteResearch use only, not for human use.
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Brief DescriptionUniPR505 is a potent EphA2 antagonist (IC50: 0.95 μM), a novel 3α-carbamoyloxy derivative with antiangiogenic properties.
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DescriptionUniPR505 (Compound 14) is an EphA2 antagonist with an IC50 of 0.95 μM. UniPR505 displays anti-angiogenic properties.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayTyrosine Kinase
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TargetEphrin Receptor
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RecptorEphrin Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2938227-14-4
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Formula Weight647.89
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Molecular FormulaC39H57N3O5
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Purity>98% (HPLC)
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Solubility——
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SMILESC[C@@]12[C@]([C@]3([C@@]([C@]4(C)[C@](CC3)(C[C@H](OC(NCC)=O)CC4)[H])(CC1)[H])[H])(CC[C@@]2([C@@H](CCC(N[C@@H](CC=5C=6C(NC5)=CC=CC6)CC(O)=O)=O)C)[H])[H]
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Incerti M, et al. Optimization of EphA2 antagonists based on a lithocholic acid core led to the identification of UniPR505, a new 3α-carbamoyloxy derivative with antiangiogenetic properties. Eur J Med Chem. 2020 Mar 1;189:112083. ?
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UniPR505
UniPR505 is a potent EphA2 antagonist (IC50: 0.95 μM), a novel 3α-carbamoyloxy derivative with antiangiogenic properties.
