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UNC2250
CAS No. 1493694-70-4
UNC2250 ( UNC2250, UNC-2250, UNC 2250 )
Catalog No. M12068 CAS No. 1493694-70-4
UNC2250 is a potent and selective Mer inhibitor with IC50 of 1.7 nM, about 160- and 60-fold selectivity over the closely related kinases Axl/Tyro3.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 34 | In Stock |
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| 5MG | 55 | In Stock |
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| 10MG | 91 | In Stock |
|
| 25MG | 174 | In Stock |
|
| 50MG | 323 | In Stock |
|
| 100MG | 480 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameUNC2250
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NoteResearch use only, not for human use.
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Brief DescriptionUNC2250 is a potent and selective Mer inhibitor with IC50 of 1.7 nM, about 160- and 60-fold selectivity over the closely related kinases Axl/Tyro3.
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DescriptionUNC2250 is a potent and selective Mer inhibitor with IC50 of 1.7 nM, about 160- and 60-fold selectivity over the closely related kinases Axl/Tyro3.
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SynonymsUNC2250, UNC-2250, UNC 2250
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PathwayTyrosine Kinase
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TargetTAM Receptor
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RecptorAXL; Mer; Tyro3
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1493694-70-4
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Formula Weight440.58
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Molecular FormulaC24H36N6O2
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Purity>98%(HPLC)
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SolubilityDMSO: 2 mg/mL warmed (4.53 mM)
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SMILESO[C@H]1CC[C@H](NC2=NC(NCCCC)=NC=C2C3=NC=C(CN4CCOCC4)C=C3)CC1
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Chemical Name(1r,4r)-4-((2-(butylamino)-5-(5-(morpholinomethyl)pyridin-2-yl)pyrimidin-4-yl)amino)cyclohexanol
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Zhang W, et al. J Med Chem. 2013, 56(23), 9683-9692.
molnova catalog
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