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Temanogrel
CAS No. 887936-68-7
Temanogrel ( APD791 )
Catalog No. M24910 CAS No. 887936-68-7
Temanogrel is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 237 | In Stock |
|
| 10MG | 354 | In Stock |
|
| 25MG | 592 | In Stock |
|
| 50MG | 843 | In Stock |
|
| 100MG | 1143 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTemanogrel
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NoteResearch use only, not for human use.
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Brief DescriptionTemanogrel is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
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DescriptionTemanogrel is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
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SynonymsAPD791
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT2A
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Research Area——
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Indication——
Chemical Information
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CAS Number887936-68-7
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Formula Weight436.5
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Molecular FormulaC24H28N4O4
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Purity>98% (HPLC)
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SolubilityDMSO:125 mg/mL (286.37 mM; Need ultrasonic)
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SMILESCn1nccc1-c(cc(cc1)NC(c2cc(OC)ccc2)=O)c1OCCN1CCOCC1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Xiong Y, et al. Discovery and structure-activity relationship of 3-methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): a highly selective 5-hydroxytryptamine2A receptor inverse agonist for the treatment of arterial thrombosis. J Med Chem. 2010 Jun 10;53(11):4412-21.
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