TP-10

CAS No. 898563-00-3

TP-10 ( —— )

Catalog No. M26489 CAS No. 898563-00-3

TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 177 Get Quote
10MG 264 Get Quote
25MG 461 Get Quote
50MG 669 Get Quote
100MG 945 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    TP-10
  • Note
    Research use only, not for human use.
  • Brief Description
    TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.
  • Description
    TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.(In Vivo):TP-10 is active in the mouse behavioral model for positive symptoms. TP-10 demonstrates good in vitro and in vivo activity with extremely high intrinsic clearance (CLint) of t>1000 mL/min/kg in mouse liver microsomes (MLM) in assay.
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    PDE
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    898563-00-3
  • Formula Weight
    460.5
  • Molecular Formula
    C26H19F3N4O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    FC(F)(F)Cn1cc(c(n1)-c1ccc(OCc2ccc3ccccc3n2)cc1)-c1ccncc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Tadros W, Boulos AL. Selective hydrogenation of ergosterol and its acetate. Helv Chim Acta. 1975 Apr 23;58(3):668-71.
molnova catalog
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