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TP-10
CAS No. 898563-00-3
TP-10 ( —— )
Catalog No. M26489 CAS No. 898563-00-3
TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 177 | Get Quote |
|
| 10MG | 264 | Get Quote |
|
| 25MG | 461 | Get Quote |
|
| 50MG | 669 | Get Quote |
|
| 100MG | 945 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameTP-10
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NoteResearch use only, not for human use.
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Brief DescriptionTP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.
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DescriptionTP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.(In Vivo):TP-10 is active in the mouse behavioral model for positive symptoms. TP-10 demonstrates good in vitro and in vivo activity with extremely high intrinsic clearance (CLint) of t>1000 mL/min/kg in mouse liver microsomes (MLM) in assay.
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Synonyms——
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PathwayAngiogenesis
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TargetPDE
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number898563-00-3
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Formula Weight460.5
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Molecular FormulaC26H19F3N4O
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Purity>98% (HPLC)
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Solubility——
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SMILESFC(F)(F)Cn1cc(c(n1)-c1ccc(OCc2ccc3ccccc3n2)cc1)-c1ccncc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Tadros W, Boulos AL. Selective hydrogenation of ergosterol and its acetate. Helv Chim Acta. 1975 Apr 23;58(3):668-71.
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