TAS6417

CAS No. 1661854-97-2

TAS6417 ( —— )

Catalog No. M23746 CAS No. 1661854-97-2

TAS6417 is an EGFR inhibitor and is an efficacious drug candidate for patients with NSCLC.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 178 In Stock
10MG 295 In Stock
25MG 597 In Stock
50MG 954 In Stock
100MG 1467 In Stock
500MG 2952 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    TAS6417
  • Note
    Research use only, not for human use.
  • Brief Description
    TAS6417 is an EGFR inhibitor and is an efficacious drug candidate for patients with NSCLC.
  • Description
    TAS6417 is an EGFR inhibitor and is an efficacious drug candidate for patients with NSCLC (IC50: ranging from 1.1-8.0 nM).
  • Synonyms
    ——
  • Pathway
    Apoptosis
  • Target
    Apoptosis
  • Recptor
    Apoptosis;EGFR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1661854-97-2
  • Formula Weight
    396.4
  • Molecular Formula
    C23H20N6O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:125 mg/mL (315.31 mM)
  • SMILES
    CC1=C[C@@H](CN2C1=C(C3=C(N=CN=C32)N)C4=CC5=CC=CC=C5N=C4)NC(=O)C=C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Hasako S, et al. TAS6417, A Novel EGFR Inhibitor Targeting Exon 20 Insertion Mutations. Mol Cancer Ther. 2018 Aug;17(8):1648-1658.
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