Seclidemstat

CAS No. 1423715-37-0

Seclidemstat ( SP-2577;SP2577 )

Catalog No. M11789 CAS No. 1423715-37-0

Seclidemstat (SP-2577, SP2577) is a potent, selectiveLSD1inhibitor with IC50 of 127 nM,reduces tumor volume in vivo.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 37 In Stock
10MG 59 In Stock
25MG 111 In Stock
50MG 177 In Stock
100MG 336 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Seclidemstat
  • Note
    Research use only, not for human use.
  • Brief Description
    Seclidemstat (SP-2577, SP2577) is a potent, selectiveLSD1inhibitor with IC50 of 127 nM,reduces tumor volume in vivo.
  • Description
    Seclidemstat (SP-2577, SP2577) is a potent, selectiveLSD1inhibitor with IC50 of 127 nM,reduces tumor volume in vivo.
  • Synonyms
    SP-2577;SP2577
  • Pathway
    Chromatin/Epigenetic
  • Target
    Histone Demethylase
  • Recptor
    LSD1
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1423715-37-0
  • Formula Weight
    450.94
  • Molecular Formula
    C20H23ClN4O4S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: Soluble ( < 1 mg/ml refers to the product slightly soluble or insoluble )
  • SMILES
    O=C(N/N=C(C1=CC(Cl)=CC=C1O)\C)C2=CC=CC(S(=O)(N3CCN(C)CC3)=O)=C2
  • Chemical Name
    N'-[(1E)-1-(5-chloro-2-hydroxyphenyl)ethylidene]-3-(4-methylpiperazine-1-sulfonyl)benzohydrazide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. PatentWO/2017/004519 A1.
molnova catalog
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