Saclofen

CAS No. 125464-42-8

Saclofen ( Saclofen )

Catalog No. M17221 CAS No. 125464-42-8

Saclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 μM).

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 110 In Stock
10MG 177 In Stock
25MG 410 In Stock
50MG 605 In Stock
100MG 860 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Saclofen
  • Note
    Research use only, not for human use.
  • Brief Description
    Saclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 μM).
  • Description
    Saclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 μM). This compound can be used to determine the functional roles for the GABAB receptor as a mediator of slow inhibitory postsynaptic potentials in the brain.
  • Synonyms
    Saclofen
  • Pathway
    Endocrinology/Hormones
  • Target
    Androgen Receptor (AR)
  • Recptor
    GABAB
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    125464-42-8
  • Formula Weight
    249.71
  • Molecular Formula
    C9H12ClNO3S
  • Purity
    98%
  • Solubility
    ——
  • SMILES
    NCC(CS(O)(=O)=O)c1ccc(Cl)cc1
  • Chemical Name
    3-Amino-2-(4-chlorophenyl)propane-1-sulfonic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Drew C A, Johnston G A R, Kerr D I B, et al. Neuroscience letters, 1990, 113(1): 107-110.
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