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STAT3-IN-1
CAS No. 2059952-75-7
STAT3-IN-1 ( —— )
Catalog No. M21979 CAS No. 2059952-75-7
STAT3-IN-1 selective and orally active inhibitor of STAT3(in HT29 and MDA-MB 231 cells, with IC50 values of 1.82 μM and 2.14 μM , respectively), induces tumor apoptosis.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 73 | Get Quote |
|
| 5MG | 120 | Get Quote |
|
| 10MG | 183 | Get Quote |
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| 25MG | 331 | Get Quote |
|
| 50MG | 496 | Get Quote |
|
| 100MG | 714 | Get Quote |
|
| 500MG | 1467 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameSTAT3-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionSTAT3-IN-1 selective and orally active inhibitor of STAT3(in HT29 and MDA-MB 231 cells, with IC50 values of 1.82 μM and 2.14 μM , respectively), induces tumor apoptosis.
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DescriptionSTAT3-IN-1 selective and orally active inhibitor of STAT3(in HT29 and MDA-MB 231 cells, with IC50 values of 1.82 μM and 2.14 μM , respectively), induces tumor apoptosis. STAT3-IN-1 ?induces tumor cells apoptosis in MDA-MB-231 cells.
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Synonyms——
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PathwayJAK/STAT Signaling
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TargetSTAT
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RecptorSTAT3
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Research Area——
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Indication——
Chemical Information
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CAS Number2059952-75-7
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Formula Weight475.53
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Molecular FormulaC28H29NO6
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Purity>98% (HPLC)
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SolubilityDMSO:125 mg/mL?(262.86 mM;?Need ultrasonic)
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SMILESCOc1cc(OC)cc(\C=C\c2ccc(NC(=O)\C=C\c3cc(OC)c(OC)c(OC)c3)cc2)c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Li S, et al. Discovery of oral-available resveratrol-caffeic acid based hybrids inhibiting acetylated and phosphorylated STAT3 protein. Eur J Med Chem. 2016 Nov 29;124:1006-1018.
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