SJ995973

CAS No. 2882065-25-8

SJ995973( —— )

Catalog No. M37131 CAS No. 2882065-25-8

SJ995973 is a highly potent bromodomain and extraterminal (BET) protein degrader and a BET PROTAC with potential anticancer activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 347 In Stock
5MG 655 In Stock
10MG 1121 In Stock
25MG 1638 In Stock
50MG 2190 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    SJ995973
  • Note
    Research use only, not for human use.
  • Brief Description
    SJ995973 is a highly potent bromodomain and extraterminal (BET) protein degrader and a BET PROTAC with potential anticancer activity.
  • Description
    SJ995973 (PROTAC) is a uniquely potent degrader ofbromodomain and extra-terminal (BET) proteins.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    PROTACs
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2882065-25-8
  • Formula Weight
    730.28
  • Molecular Formula
    C37H40ClN7O5S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (136.93 mM; Ultrasonic )
  • SMILES
    CC=1C2=C(N3C([C@H](CC(NCCCCCNC(COC4=CC=C(C=C4)C5C(=O)NC(=O)CC5)=O)=O)N=C2C6=CC=C(Cl)C=C6)=NN=C3C)SC1C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Min J, et al. Phenyl-Glutarimides: Alternative Cereblon Binders for the Design of PROTACs. Angew Chem Int Ed Engl. 2021 Dec 13;60(51):26663-26670. ?
molnova catalog
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