SGC-GAK-1

CAS No. 2226517-76-4

SGC-GAK-1 ( —— )

Catalog No. M19961 CAS No. 2226517-76-4

SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 65 In Stock
10MG 110 In Stock
25MG 222 In Stock
50MG 357 In Stock
100MG 530 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    SGC-GAK-1
  • Note
    Research use only not for human use.
  • Brief Description
    SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).
  • Description
    SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GAK
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2226517-76-4
  • Formula Weight
    389.24
  • Molecular Formula
    C18H17BrN2O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 40 mg/mL;Ethanol: 15 mg/mL
  • SMILES
    COc1cc(Nc2ccnc3ccc(Br)cc23)cc(OC)c1OC
  • Chemical Name
    6-Bromo-N-(345-trimethoxyphenyl)quinolin-4-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Asquith CRM et al. SGC-GAK-1: A Chemical Probe for Cyclin G Associated Kinase (GAK). J Med Chem. 2019 Feb 26.
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