SB273005

CAS No. 205678-31-5

SB273005( SB-273005 | SB 273005 | SB273005 )

Catalog No. M17422 CAS No. 205678-31-5

SB273005 is a potent integrin inhibitor with Ki of 1.2 nM and 0.3 nM for αvβ3 receptor and αvβ5 receptor, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 561 Get Quote
25MG 1457 Get Quote
50MG 1782 Get Quote
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Biological Information

  • Product Name
    SB273005
  • Note
    Research use only, not for human use.
  • Brief Description
    SB273005 is a potent integrin inhibitor with Ki of 1.2 nM and 0.3 nM for αvβ3 receptor and αvβ5 receptor, respectively.
  • Description
    SB-273005 is an inhibitor of integrin αvβ3.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    SB-273005 | SB 273005 | SB273005
  • Pathway
    Tyrosine Kinase
  • Target
    Src
  • Recptor
    αVβ3 integrin| αVβ5 integrin
  • Research Area
    Inflammation/Immunology
  • Indication
    ——

Chemical Information

  • CAS Number
    205678-31-5
  • Formula Weight
    451.44
  • Molecular Formula
    C22H24F3N3O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CNC1=CC=CC(CCOC2=CC=C3C[C@@H](CC(O)=O)C(=O)N(CC(F)(F)F)CC3=C2)=N1
  • Chemical Name
    2-[(4S)-8-[2-[6-(Methylamino)pyridin-2-yl]ethoxy]-3-oxo-2-(2,2,2-trifluoroethyl)-4,5-dihydro-1H-2-benzazepin-4-yl]acetic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Miller WH, et al. J Med Chem. 2000, 43(1), 22-26.
molnova catalog
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