RN-1747
CAS No. 1024448-59-6
RN-1747 ( —— )
Catalog No. M26807 CAS No. 1024448-59-6
RN-1747 is a selective transient receptor potential cation channel subfamily V member 4 agonists (EC50: hTRPV4 of 0.77 μM, mTRPV4 of 4.0 μM, and rTRPV4 of 4.1 μM). RN-1747 also antagonizes TRPM8 (IC50: 4 μM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 34 | Get Quote |
|
5MG | 55 | Get Quote |
|
10MG | 104 | Get Quote |
|
25MG | 192 | Get Quote |
|
50MG | 312 | Get Quote |
|
100MG | 500 | Get Quote |
|
200MG | 713 | Get Quote |
|
500MG | 1062 | Get Quote |
|
1G | Get Quote | Get Quote |
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Biological Information
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Product NameRN-1747
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NoteResearch use only, not for human use.
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Brief DescriptionRN-1747 is a selective transient receptor potential cation channel subfamily V member 4 agonists (EC50: hTRPV4 of 0.77 μM, mTRPV4 of 4.0 μM, and rTRPV4 of 4.1 μM). RN-1747 also antagonizes TRPM8 (IC50: 4 μM).
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DescriptionRN-1747 is a selective transient receptor potential cation channel subfamily V member 4 agonists (EC50: hTRPV4 of 0.77 μM, mTRPV4 of 4.0 μM, and rTRPV4 of 4.1 μM). RN-1747 also antagonizes TRPM8 (IC50: 4 μM).
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number1024448-59-6
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Formula Weight395.9
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Molecular FormulaC17H18ClN3O4S
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Purity>98% (HPLC)
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Solubility——
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SMILES[O-][N+](=O)c1cc(Cl)ccc1S(=O)(=O)N1CCN(Cc2ccccc2)CC1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Weisong Zhao, et al. Biodegradation of thifensulfuron-methyl by Ochrobactrum sp. in liquid medium and soil. Biotechnol Lett. 2015 Jul;37(7):1385-92.
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