Cart
sales@molnova.com
RK-287107
CAS No. 2171386-10-8
RK-287107 ( —— )
Catalog No. M23984 CAS No. 2171386-10-8
RK-287107 is an effective and specific inhibitor of tankyrase (IC50s: 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 177 | In Stock |
|
| 10MG | 282 | In Stock |
|
| 25MG | 531 | In Stock |
|
| 50MG | 767 | In Stock |
|
| 100MG | 1053 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameRK-287107
-
NoteResearch use only, not for human use.
-
Brief DescriptionRK-287107 is an effective and specific inhibitor of tankyrase (IC50s: 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively).
-
DescriptionRK-287107 is an effective and specific inhibitor of tankyrase (IC50s: 14.3 and 10.6 nM for tankyrase-1 and tankyrase-2, respectively).
-
Synonyms——
-
PathwayOthers
-
TargetOther Targets
-
Recptortankyrase 1;tankyrase 2
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number2171386-10-8
-
Formula Weight416.5
-
Molecular FormulaC22H26F2N4O2
-
Purity>98% (HPLC)
-
SolubilityDMSO:120 mg/mL (288.14 mM; Need ultrasonic)
-
SMILESOCCN(C1)c2cc(F)cc(F)c2C1(CC1)CCN1C(N1)=NC(CCCC2)=C2C1=O
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Mizutani A, et al. RK-287107, a potent and specific tankyrase inhibitor, blocks colorectal cancer cell growth in a preclinical model. Cancer Sci. 2018 Dec;109(12):4003-4014.
molnova catalog
related products
-
Hydroxy-PEG12-Boc
Hydroxy-PEG12-Boc is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs.
-
Thalidomide-NH-PEG1-...
Thalidomide-NH-PEG1-NH2 hydrochloride is a synthetic E3 ligase ligand-linker conjugate that incorporates the Thalidomide-based cereblon ligand and a linker.
-
20-DEOXYINGENOL
20-DEOXYINGENOL is a natual product.
