Pyributicarb

CAS No. 88678-67-5

Pyributicarb ( TSH-888 )

Catalog No. M20997 CAS No. 88678-67-5

Pyributicarb is a potent activator of both CYP3A4 gene and human pregnane X receptor (hPXR).?

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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50MG 65 Get Quote
100MG 95 Get Quote
200MG 140 Get Quote
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Biological Information

  • Product Name
    Pyributicarb
  • Note
    Research use only not for human use.
  • Brief Description
    Pyributicarb is a potent activator of both CYP3A4 gene and human pregnane X receptor (hPXR).?
  • Description
    Pyributicarb is a potent activator of both CYP3A4 gene and human pregnane X receptor (hPXR).?
  • Synonyms
    TSH-888
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    P450
  • Recptor
    CYP3A4
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    88678-67-5
  • Formula Weight
    330.44
  • Molecular Formula
    C18H22N2O2S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:100 mg/mL (302.63 mM)
  • SMILES
    COc1cccc(N(C)C(=S)Oc2cccc(C(C)(C)C)c2)n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Matsubara T Noracharttiyapot W Toriyabe T et al. Assessment of Human Pregnane X Receptor Involvement in Pesticide-Mediated Activation of CYP3A4 Gene[J]. Drug Metabolism and Disposition 2007 35(5):728-733.
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