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Pipequaline

CAS No. 77472-98-1

Pipequaline( PK-8165 | PK8165 | PK 8165 )

Catalog No. M15927 CAS No. 77472-98-1

A clinically-effective anxiolytic that acts as a non-selective partial agonist of benzodiazepine receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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25MG 113 In Stock
50MG 211 In Stock
100MG 365 In Stock
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Biological Information

  • Product Name
    Pipequaline
  • Note
    Research use only, not for human use.
  • Brief Description
    A clinically-effective anxiolytic that acts as a non-selective partial agonist of benzodiazepine receptor.
  • Description
    A clinically-effective anxiolytic that acts as a non-selective partial agonist of benzodiazepine receptor; exerts a partial suppression of activations by kainate, glutamate and acetylcholine in rats, also reduces the neuronal activation by kainate.
  • In Vitro
    ——
  • In Vivo
    Intravenously administered pipequaline exerts a partial suppression of activations by kainate, glutamate and acetylcholine. Microiontophoretic applications of pipequaline reduces the neuronal activation by kainate. Pipequaline produces dose-related decreases in motor activity. Pipequaline produces significant dose-related decreases in the number of head-dips made.
  • Synonyms
    PK-8165 | PK8165 | PK 8165
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    GAT
  • Recptor
    GABAA
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    77472-98-1
  • Formula Weight
    316.4394
  • Molecular Formula
    C22H24N2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 32 mg/mL
  • SMILES
    C1CNCCC1CCC2=CC(=NC3=CC=CC=C32)C4=CC=CC=C4
  • Chemical Name
    Quinoline, 2-phenyl-4-[2-(4-piperidinyl)ethyl]-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. File SE. Br J Pharmacol. 1983 May;79(1):219-23. 2. Gee KW, et al. Brain Res. 1983 Mar 28;264(1):168-72. 3. Debonnel G, et al. Neuropharmacology. 1987 Sep;26(9):1337-42.
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