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Pimethixene

CAS No. 314-03-4

Pimethixene ( Pimetixene; Calmixen )

Catalog No. M24244 CAS No. 314-03-4

Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 43 In Stock
5MG 64 In Stock
10MG 91 In Stock
25MG 162 In Stock
50MG 240 In Stock
100MG 357 In Stock
200MG 534 In Stock
500MG 854 In Stock
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Biological Information

  • Product Name
    Pimethixene
  • Note
    Research use only, not for human use.
  • Brief Description
    Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
  • Description
    Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
  • Synonyms
    Pimetixene; Calmixen
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT2A Receptor;5-HT2B Receptor;5-HT2C Receptor;H1 receptor;5-HT1A Receptor;D2 receptor;DD4.4 receptor;M1 receptor;M2 receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    314-03-4
  • Formula Weight
    293.4
  • Molecular Formula
    C19H19NS
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CN(CC1)CCC1=C1c(cccc2)c2Sc2c1cccc2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Schmitz B, et al. BF-1--a novel selective 5-HT2B receptor antagonist blocking neurogenic dural plasma protein extravasation in guinea pigs. Eur J Pharmacol. 2015 Mar 15;751:73-80.
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