PTGR2-IN-22

CAS No. 349093-44-3

PTGR2-IN-22 ( —— )

Catalog No. M22891 CAS No. 349093-44-3

PTGR2-IN-22 is a potent inhibito of PTGR2r(IC50 : 0.7 μM). It increases 15-keto-PGE2-dependent PPARγ transcriptional activity in PTGR2-transfected HEK293T cells.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 147 Get Quote
10MG 222 Get Quote
25MG 410 Get Quote
50MG 605 Get Quote
100MG 860 Get Quote
500MG 1728 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    PTGR2-IN-22
  • Note
    Research use only, not for human use.
  • Brief Description
    PTGR2-IN-22 is a potent inhibito of PTGR2r(IC50 : 0.7 μM). It increases 15-keto-PGE2-dependent PPARγ transcriptional activity in PTGR2-transfected HEK293T cells.
  • Description
    PTGR2-IN-22 is a potent inhibito of PTGR2r(IC50 : 0.7 μM). It increases 15-keto-PGE2-dependent PPARγ transcriptional activity in PTGR2-transfected HEK293T cells.
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    PTGR2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    349093-44-3
  • Formula Weight
    310.39
  • Molecular Formula
    C19H22N2O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:100 mg/mL (322.18 mM; Need ultrasonic)
  • SMILES
    COC1=CC=CC=C1N2CCN(C(CC3=CC=CC=C3)=O)CC2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Parker CG, et al. Ligand and Target Discovery by Fragment-Based Screening in Human Cells. Cell. 2017;168(3):527-541.e29.
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