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PSI-421
CAS No. 1067186-56-4
PSI-421( PSI 421 | PSI421 )
Catalog No. M10287 CAS No. 1067186-56-4
A potent, orally bioavailable P-selectin inhibitor with improved pharmacokinetic properties and oral efficacy in models of vascular injury.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NamePSI-421
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, orally bioavailable P-selectin inhibitor with improved pharmacokinetic properties and oral efficacy in models of vascular injury.
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DescriptionA potent, orally bioavailable P-selectin inhibitor with improved pharmacokinetic properties and oral efficacy in models of vascular injury.
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In Vitro——
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In Vivo——
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SynonymsPSI 421 | PSI421
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetSelectin
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RecptorSelectin
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Research Area——
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Indication——
Chemical Information
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CAS Number1067186-56-4
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Formula Weight407.773
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Molecular FormulaC20H13ClF3NO3
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Purity>98% (HPLC)
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Solubility——
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SMILESC1CC1(C2=CC=C(C=C2)Cl)C3=C(C(=C4C=CC=C(C4=N3)C(F)(F)F)C(=O)O)O
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Chemical Name2-[1-(4-chlorophenyl)cyclopropyl]-3-hydroxy-8-(trifluoromethyl)quinoline-4-carboxylic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Huang A, et al. J Med Chem. 2010 Aug 26;53(16):6003-17.
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