Cart
sales@molnova.com
PF-06882961
CAS No. 2230198-02-2
PF-06882961( —— )
Catalog No. M22917 CAS No. 2230198-02-2
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist. PF-06882961 shows mild to moderate damage to the heart, moderate to severe effects on the thymus gland (which helps with managing infection), mild to moderate stomach ulcers at the highest dose level given in the rat.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 201 | In Stock |
|
| 10MG | 314 | In Stock |
|
| 25MG | 602 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NamePF-06882961
-
NoteResearch use only, not for human use.
-
Brief DescriptionPF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist. PF-06882961 shows mild to moderate damage to the heart, moderate to severe effects on the thymus gland (which helps with managing infection), mild to moderate stomach ulcers at the highest dose level given in the rat.
-
DescriptionPF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist. PF-06882961 shows mild to moderate damage to the heart, moderate to severe effects on the thymus gland (which helps with managing infection), mild to moderate stomach ulcers at the highest dose level given in the rat.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayGPCR/G Protein
-
TargetGlucagon Receptor
-
RecptorGLP-1
-
Research AreaMetabolism
-
IndicationDiabetes Mellitus, Type 2
Chemical Information
-
CAS Number2230198-02-2
-
Formula Weight555.6
-
Molecular FormulaC31H30FN5O4
-
Purity>98% (HPLC)
-
SolubilityDMSO:125 mg/mL (224.98 mM; Need ultrasonic)
-
SMILESOC(C1=CC=C(N=C(CN2CCC(C3=NC(OCC4=CC=C(C#N)C=C4F)=CC=C3)CC2)N5C[C@H]6OCC6)C5=C1)=O
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. 20th SCI/RSC Medicinal Chemistry Symposium.
molnova catalog
related products
-
NNC 92-1687
NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.
-
GLP-2(1-33)(human)
GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.
-
NNC-0640
NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
