PF-06869206

CAS No. 2227425-05-8

PF-06869206 ( —— )

Catalog No. M24011 CAS No. 2227425-05-8

PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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2MG 31 In Stock
5MG 50 In Stock
10MG 87 In Stock
25MG 192 In Stock
50MG 332 In Stock
100MG 494 In Stock
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Biological Information

  • Product Name
    PF-06869206
  • Note
    Research use only, not for human use.
  • Brief Description
    PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).
  • Description
    PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).
  • Synonyms
    ——
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    Sodium Channel
  • Recptor
    SLC34A1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2227425-05-8
  • Formula Weight
    374.8
  • Molecular Formula
    C15H14ClF3N4O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:120 mg/mL (320.22 mM)
  • SMILES
    CC1=C(C2=C(N1)C(=C(C(=N2)C(F)(F)F)C#N)N3CCO[C@@H](C3)CO)Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Filipski KJ, et al. Discovery of Orally Bioavailable Selective Inhibitors of the Sodium-Phosphate Cotransporter NaPi2a (SLC34A1). ACS Med Chem Lett. 2018 Apr 12;9(5):440-445.
molnova catalog
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