PF-06821497

CAS No. 1844849-10-0

PF-06821497 ( —— )

Catalog No. M26370 CAS No. 1844849-10-0

PF-06821497 is a selective inhibitor of EZH2 with significant tumor growth inhibition.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 393 Get Quote
10MG 581 Get Quote
25MG 888 Get Quote
50MG 1242 Get Quote
100MG 1674 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    PF-06821497
  • Note
    Research use only, not for human use.
  • Brief Description
    PF-06821497 is a selective inhibitor of EZH2 with significant tumor growth inhibition.
  • Description
    PF-06821497 is a selective inhibitor of EZH2 with significant tumor growth inhibition.(In Vivo):The tumor regression effect of PF-06821497 can be sustained for another 40 days.
  • Synonyms
    ——
  • Pathway
    Chromatin/Epigenetic
  • Target
    Histone Demethylase
  • Recptor
    Apoptosis; Autophagy
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1844849-10-0
  • Formula Weight
    467.3
  • Molecular Formula
    C22H24Cl2N2O5
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CO[C@H](C1COC1)c1cc(Cl)c2CCN(Cc3c(OC)cc(C)[nH]c3=O)C(=O)c2c1Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Greim H, Saltmiras D, Mostert V, Strupp C. Evaluation of carcinogenic potential of the herbicide glyphosate, drawing on tumor incidence data from fourteen chronic/carcinogenicity rodent studies. Crit Rev Toxicol. 2015 Mar;45(3):185-208.
molnova catalog
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