PF-04995274
CAS No. 1331782-27-4
PF-04995274 ( PF-4995274;TBPT )
Catalog No. M11321 CAS No. 1331782-27-4
PF-04995274 (TBPT) is a novel potent, sellective, partial agonist of 5-HT4 receptor under investigation for neurological disorders.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 61 | Get Quote |
|
10MG | 113 | Get Quote |
|
25MG | 186 | Get Quote |
|
50MG | 332 | Get Quote |
|
100MG | 478 | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePF-04995274
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NoteResearch use only, not for human use.
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Brief DescriptionPF-04995274 (TBPT) is a novel potent, sellective, partial agonist of 5-HT4 receptor under investigation for neurological disorders.
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DescriptionPF-04995274 (TBPT) is a novel potent, sellective, partial agonist of 5-HT4 receptor under investigation for neurological disorders.Alzheimer Disease Phase 1 Discontinued
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SynonymsPF-4995274;TBPT
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT Receptor
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Research AreaNeurological Disease
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IndicationAlzheimer Disease
Chemical Information
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CAS Number1331782-27-4
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Formula Weight432.52
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Molecular FormulaC23H32N2O6
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Purity>98% (HPLC)
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Solubility——
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SMILESC1CN(CCC1COC2=NOC3=C2C(=CC=C3)OC4CCOC4)CC5(CCOCC5)O
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Chemical Name(R)-4-((4-(((4-(Tetrahydrofuran-3-yloxy)-1,2-benzisoxazol-3-yl)oxy)methyl)piperidin-1-yl)methyl)tetrahydro-2H-pyran-4-ol
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Sawant-Basak A, et al. J Pharm Sci. 2013 Sep;102(9):3277-93.
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