Cart
sales@molnova.com
Home - Products - Endocrinology/Hormones - 5-HT Receptor - PF-03246799

PF-03246799

CAS No. 1065110-62-4

PF-03246799 ( PF 03246799;PF03246799;PF-3246799 )

Catalog No. M10282 CAS No. 1065110-62-4

A potent and selective 5-HT2C receptor agonist with EC50 of 190 nM, with excellent selectivity for 5-HT2C over 5-HT2A.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 873 Get Quote
50MG 1782 Get Quote
100MG 2250 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote
Group Booking Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    PF-03246799
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent and selective 5-HT2C receptor agonist with EC50 of 190 nM, with excellent selectivity for 5-HT2C over 5-HT2A.
  • Description
    A potent and selective 5-HT2C receptor agonist with EC50 of 190 nM, with excellent selectivity for 5-HT2C over 5-HT2A; has minimal activation at either the 5-HT(2A) or 5-HT(2B) receptors, demonstrates robust efficacy in preclinical canine model of stress urinary incontinence (SUI) and attractive pharmacokinetic and safety properties.
  • Synonyms
    PF 03246799;PF03246799;PF-3246799
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1065110-62-4
  • Formula Weight
    239.32
  • Molecular Formula
    C15H17N3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C12=NC(CC3=CC=CC=C3)=NC=C1CCNCC2
  • Chemical Name
    2-benzyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Andrews MD, et al. Bioorg Med Chem Lett. 2011 May 1;21(9):2715-20.
2. Dvorak CA, et al. ACS Med Chem Lett. 2015 Jul 20;6(9):1015-8.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • 2-Methyl-5-HT

    2-Methyl-5-HT is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.

  • Sodium ascorbate

    Sodium Ascorbate is a more bioavailable form of vitamin C that is an alternative to taking ascorbic acid as a supplement.

  • Promethazine

    Tafluprost(AFP-168) is an anti-glaucoma prostaglandin (PG) analog.

Sign In Join Free