
PF-03246799
CAS No. 1065110-62-4
PF-03246799( PF 03246799 | PF03246799 | PF-3246799 )
Catalog No. M10282 CAS No. 1065110-62-4
A potent and selective 5-HT2C receptor agonist with EC50 of 190 nM, with excellent selectivity for 5-HT2C over 5-HT2A.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
5MG | 873 | Get Quote |
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50MG | 1782 | Get Quote |
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100MG | 2250 | Get Quote |
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200MG | Get Quote | Get Quote |
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500MG | Get Quote | Get Quote |
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1G | Get Quote | Get Quote |
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Biological Information
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Product NamePF-03246799
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NoteResearch use only, not for human use.
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Brief DescriptionA potent and selective 5-HT2C receptor agonist with EC50 of 190 nM, with excellent selectivity for 5-HT2C over 5-HT2A.
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DescriptionA potent and selective 5-HT2C receptor agonist with EC50 of 190 nM, with excellent selectivity for 5-HT2C over 5-HT2A; has minimal activation at either the 5-HT(2A) or 5-HT(2B) receptors, demonstrates robust efficacy in preclinical canine model of stress urinary incontinence (SUI) and attractive pharmacokinetic and safety properties.
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In Vitro——
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In Vivo——
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SynonymsPF 03246799 | PF03246799 | PF-3246799
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number1065110-62-4
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Formula Weight239.322
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Molecular FormulaC15H17N3
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Purity>98% (HPLC)
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Solubility——
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SMILESC12=NC(CC3=CC=CC=C3)=NC=C1CCNCC2
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Chemical Name2-benzyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference



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