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PAP-1
CAS No. 870653-45-5
PAP-1 ( 5-(4-Phenoxybutoxy)psoralen )
Catalog No. M24882 CAS No. 870653-45-5
PAP-1 is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 51 | In Stock |
|
| 5MG | 73 | In Stock |
|
| 10MG | 124 | In Stock |
|
| 25MG | 276 | In Stock |
|
| 50MG | 492 | In Stock |
|
| 100MG | 520 | In Stock |
|
| 200MG | 744 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePAP-1
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NoteResearch use only, not for human use.
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Brief DescriptionPAP-1 is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).
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DescriptionPAP-1 is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).
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Synonyms5-(4-Phenoxybutoxy)psoralen
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PathwayCell Cycle/DNA Damage
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TargetPotassium Channel
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RecptorKv1.3 channels
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Research Area——
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Indication——
Chemical Information
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CAS Number870653-45-5
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Formula Weight350.4
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Molecular FormulaC21H18O5
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Purity>98% (HPLC)
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SolubilityDMSO:48 mg/mL (137 mM; Need ultrasonic);Water:Insoluble
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SMILESO=C(C=C1)Oc2c1c(OCCCCOc1ccccc1)c(cco1)c1c2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Schmitz A, et al. Design of PAP-1, a selective small molecule Kv1.3 blocker, for the suppression of effector memory T cells in autoimmune diseases. Mol Pharmacol. 2005 Nov;68(5):1254-70.
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