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OXFBD04
CAS No. 2231747-03-6
OXFBD04 ( —— )
Catalog No. M26352 CAS No. 2231747-03-6
OXFBD04 is a potent and selective inhibitor of BRD4(IC50 of 166 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 152 | Get Quote |
|
| 5MG | 260 | Get Quote |
|
| 10MG | 444 | Get Quote |
|
| 25MG | 712 | Get Quote |
|
| 50MG | 1008 | Get Quote |
|
| 100MG | 1341 | Get Quote |
|
| 500MG | 2673 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameOXFBD04
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NoteResearch use only, not for human use.
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Brief DescriptionOXFBD04 is a potent and selective inhibitor of BRD4(IC50 of 166 nM).
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DescriptionOXFBD04 is a potent and selective inhibitor of BRD4(IC50 of 166 nM).(In Vitro):OXFBD04 (0.01-100 μM) inhibits the cell growth of cancer cell lines. In MCF7 breast cancer cells, OXFBD04 (10?μM) induces MYC suppression.(In Vivo):OXFBD04 has optimized physicochemical properties (LE = 0.43; LLE = 5.74; SFI = 5.96), and greater metabolic stability (t1/2 = 388?min, CLint = 3.57 μL/min/mg).
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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RecptorAnti-infection; Antibacterial; Antibiotic; α-glucosidase
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Research Area——
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Indication——
Chemical Information
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CAS Number2231747-03-6
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Formula Weight296.3
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Molecular FormulaC17H16N2O3
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Purity>98% (HPLC)
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Solubility——
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SMILESCc1noc(C)c1-c1cc(O)cc(c1)C(O)c1cccnc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Nishida M, Murakawa T, Kamimura T, Okada N, Sakamoto H, Fukada S, Nakamoto S, Yokota Y, Miki K. In vitro and in vivo evaluation of ceftezole, a new cephalosporin derivative. Antimicrob Agents Chemother. 1976 Jul;10(1):1-13.
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