
Nomegestrol
CAS No. 58691-88-6
Nomegestrol( —— )
Catalog No. M33634 CAS No. 58691-88-6
Nomegestrol (TX 066 free base) is an orally available, selective and potent full agonist of the progesterone receptor with potent anti-estrogenic, partial anti-androgenic and anti-gonadotropic activity.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
2MG | 316 | Get Quote |
![]() ![]() |
500MG | Get Quote | Get Quote |
![]() ![]() |
1G | Get Quote | Get Quote |
![]() ![]() |
Biological Information
-
Product NameNomegestrol
-
NoteResearch use only, not for human use.
-
Brief DescriptionNomegestrol (TX 066 free base) is an orally available, selective and potent full agonist of the progesterone receptor with potent anti-estrogenic, partial anti-androgenic and anti-gonadotropic activity.
-
DescriptionNomegestrol is a potent and orally available progestin, acts as a selective full progesterone receptor agonist, with a Kd of 5.44 nM for rat uterine progesterone receptor, and has moderate antiandrogenic activity and strong antiestrogenic activity.
-
In VitroNomegestrol is a progestin, has high binding affinity at progesterone receptor, with a Kd of 5.44 nM for rat uterine progesterone receptor. Nomegestrol acetate (NOMAC) is a higly selective progesterone receptor full agonist, but shows no or little binding affinity at other steroid receptors, such as the androgen and glucocorticoid receptors. Nomegestrol acetate has moderate antiandrogenic activity and strong antiestrogenic activity.
-
In Vivo——
-
Synonyms——
-
PathwayNuclear Receptor/Transcription Factor
-
TargetProgesterone Receptor
-
RecptorProgesterone Receptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number58691-88-6
-
Formula Weight328.45
-
Molecular FormulaC21H28O3
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESC[C@@]12[C@]([C@]3([C@@]([C@@]4(C(C(C)=C3)=CC(=O)CC4)[H])(CC1)[H])[H])(CC[C@@]2(C(C)=O)O)[H]
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Duc I, et al. Interaction of [3H]nomegestrol acetate with cytosolic progesterone receptors from the rat uterus. Steroids. 1991 Jun;56(6):325-8.?
molnova catalog



related products
-
Norethindrone acetat...
Norethindrone acetate (19-Norethindroneacetate) is an oestrogen with inhibitory effects on adolescent menstruation and hepatic adenomas and is often used in combination with progestins in the study of endometriosis.
-
Nomegestrol acetate
Nomegestrol acetate is a widely used progestin-like drugwhich is characterized as a full agonist at the progesterone receptor.
-
Nomegestrol
Nomegestrol (TX 066 free base) is an orally available, selective and potent full agonist of the progesterone receptor with potent anti-estrogenic, partial anti-androgenic and anti-gonadotropic activity.