Cart
sales@molnova.com
N-Desmethyl-Apalutamide
CAS No. 1332391-11-3
N-Desmethyl-Apalutamide ( N-Desmethyl Apalutamide )
Catalog No. M26314 CAS No. 1332391-11-3
N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 410 | Get Quote |
|
| 10MG | 591 | Get Quote |
|
| 25MG | 888 | Get Quote |
|
| 50MG | 1224 | Get Quote |
|
| 100MG | 1647 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameN-Desmethyl-Apalutamide
-
NoteResearch use only, not for human use.
-
Brief DescriptionN-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
-
DescriptionN-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
-
SynonymsN-Desmethyl Apalutamide
-
PathwayMetabolic Enzyme/Protease
-
TargetP450
-
RecptorCYP2C9; HIV
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number1332391-11-3
-
Formula Weight463.4
-
Molecular FormulaC20H13F4N5O2S
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESNC(=O)c1ccc(cc1F)N1C(=S)N(C(=O)C11CCC1)c1cnc(C#N)c(c1)C(F)(F)F
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Chen DF, et al. Anti-AIDS agents--XXVI. Structure-activity correlations of gomisin-G-related anti-HIV lignans from Kadsura interior and of related synthetic analogues. Bioorg Med Chem. 1997 Aug;5(8):1715-23.
molnova catalog
related products
-
7-Hydroxyflavone
7-Hydroxyflavone is a potent inhibitor of CYP1A1 with a Ki value of 0.015 μM and exhibits 6-fold greater selectivity for CYP1A1 over CYP1A2.with anti-inflammatory activity.
-
1-Aminobenzotriazole
1-Aminobenzotriazole (ABT) is a non-specific cytochrome P450 (CYP) inhibitor.
-
Liarozole
Liarozole is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase).
