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Liarozole

CAS No. 115575-11-6

Liarozole ( R75251 dihydrochloride )

Catalog No. M23335 CAS No. 115575-11-6

Liarozole is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase).

Purity : >98% (HPLC)

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Size	Price / USD	Stock	Quantity
5MG	178	In Stock
10MG	295	In Stock
25MG	502	In Stock
50MG	709	In Stock
100MG	1008	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

Liarozole
Note

Research use only, not for human use.
Brief Description

Liarozole is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase).
Description

Liarozole is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase).Liarozole dihydrochloride is an imidazole derivative;?it is being investigated as a non-hormonal agent in prostate cancer and in the treatment of various other cancers and skin disorders.?
Synonyms

R75251 dihydrochloride
Pathway

Metabolic Enzyme/Protease
Target

P450
Recptor

CYP450
Research Area

——
Indication

——

Chemical Information

CAS Number

115575-11-6
Formula Weight

308.8
Molecular Formula

C17H13ClN4
Purity

>98% (HPLC)
Solubility

DMSO:10 mM
SMILES

ClC1=CC(C(C2=CC=C3NC=NC3=C2)N4C=CN=C4)=CC=C1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Bryson HM, et al. Liarozole. Drugs Aging. 1996 Dec;9(6):478-84; discussion 485.

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