Mizolastine
CAS No. 108612-45-9
Mizolastine ( SL 85.0324; Mistalin; Mistamine; Mizolastina )
Catalog No. M10337 CAS No. 108612-45-9
Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
25MG | 48 | In Stock |
|
50MG | 61 | In Stock |
|
100MG | 87 | In Stock |
|
200MG | 168 | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameMizolastine
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NoteResearch use only, not for human use.
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Brief DescriptionMizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
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DescriptionMizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
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SynonymsSL 85.0324; Mistalin; Mistamine; Mizolastina
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorH1 receptor
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number108612-45-9
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Formula Weight432.49
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Molecular FormulaC24H25FN6O
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Purity>98%(HPLC)
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SolubilityEthanol: <1 mg/mL warmed (<1 mM); Water: <1 mg/mL (<1 mM); DMSO: <1 mg/mL (<1 mM)
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SMILESO=C1NC(N(C2CCN(C3=NC4=CC=CC=C4N3CC5=CC=C(F)C=C5)CC2)C)=NC=C1
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Chemical Name2-((1-(1-(p-Fluorobenzyl)-2-benzimidazolyl)-4-piperidyl)methylamino)-4(3H)-pyrimidinone
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Brostoff J, et al.Allergy. 1996 May; 51(5):320-5.
molnova catalog
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