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MZ-242
CAS No. 1862238-01-4
MZ-242 ( MZ242;MZ242 )
Catalog No. M12877 CAS No. 1862238-01-4
A novel potent, selective Sirt2 inhibitor with IC50 of 0.118 uM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 963 | Get Quote |
|
| 50MG | 1962 | Get Quote |
|
| 100MG | 2520 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameMZ-242
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NoteResearch use only, not for human use.
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Brief DescriptionA novel potent, selective Sirt2 inhibitor with IC50 of 0.118 uM.
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DescriptionA novel potent, selective Sirt2 inhibitor with IC50 of 0.118 uM; displays no inhibitory activity against Sirt1 and Sirt 3 (IC50>100 uM).
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SynonymsMZ242;MZ242
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PathwayChromatin/Epigenetic
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TargetSirtuin
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RecptorSirtuin
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Research Area——
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Indication——
Chemical Information
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CAS Number1862238-01-4
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Formula Weight525.65
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Molecular FormulaC24H27N7O3S2
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(NC1=NC=C(CC2=CC=CC(OCC3=CN(CCOC)N=N3)=C2)S1)CSC4=NC(C)=CC(C)=N4
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Chemical Name2-((4,6-dimethylpyrimidin-2-yl)thio)-N-(5-(3-((1-(2-methoxyethyl)-1H-1,2,3-triazol-4-yl)methoxy)benzyl)thiazol-2-yl)acetamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Szabó A, et al. Sci Rep. 2017 Dec 6;7(1):17070.
2. Schiedel M, et al. Angew Chem Int Ed Engl. 2016 Feb 5;55(6):2252-6.
2. Schiedel M, et al. Angew Chem Int Ed Engl. 2016 Feb 5;55(6):2252-6.
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