MS436
CAS No. 1395084-25-9
MS436 ( MS436; MS-436; MS 436 )
Catalog No. M11651 CAS No. 1395084-25-9
MS436 is a diazobenzene-based small-molecule inhibitor for the BRD4 bromodomains with a Ki value of 30-50 nM.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 33 | In Stock |
|
5MG | 53 | In Stock |
|
10MG | 95 | In Stock |
|
25MG | 183 | In Stock |
|
50MG | 327 | In Stock |
|
100MG | 478 | In Stock |
|
500MG | 1035 | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameMS436
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NoteResearch use only, not for human use.
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Brief DescriptionMS436 is a diazobenzene-based small-molecule inhibitor for the BRD4 bromodomains with a Ki value of 30-50 nM.
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DescriptionMS436 is a diazobenzene-based small-molecule inhibitor for the BRD4 bromodomains with a Ki value of 30-50 nM.
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SynonymsMS436; MS-436; MS 436
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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RecptorBRD4 (1); BRD4 (2)
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number1395084-25-9
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Formula Weight383.42
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Molecular FormulaC18H17N5O3S
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Purity>98%(HPLC)
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SolubilityEthanol: 1 mg/mL warmed (2.6 mM); DMSO: 55 mg/mL (143.44 mM)
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SMILESO=S(C1=CC=C(/N=N/C2=CC(C)=C(O)C=C2N)C=C1)(NC3=NC=CC=C3)=O
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Chemical Name(E)-4-[2-(2-Amino-4-hydroxy-5-methylphenyl)diazenyl]-N-2-pyridinylbenzenesulfonamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Zhang G, et al. J Med Chem. 2013 Nov 27;56(22):9251-64.
molnova catalog
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