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MS012
CAS No. 2089617-83-2
MS012( MS 012 )
Catalog No. M13271 CAS No. 2089617-83-2
MS012 is a potent and selective inhibitor of G9a-Like Protein (GLP) lysine methyltransferase with IC50 of 7 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameMS012
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NoteResearch use only, not for human use.
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Brief DescriptionMS012 is a potent and selective inhibitor of G9a-Like Protein (GLP) lysine methyltransferase with IC50 of 7 nM.
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DescriptionMS012 is a potent and selective inhibitor of G9a-Like Protein (GLP) lysine methyltransferase with IC50 of 7 nM, shows >30-fold selectivity for GLP over G9a and other methyltransferases.
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In Vitro——
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In Vivo——
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SynonymsMS 012
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorHMTase
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Research Area——
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Indication——
Chemical Information
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CAS Number2089617-83-2
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Formula Weight401.555
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Molecular FormulaC22H35N5O2
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Purity>98% (HPLC)
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Solubility——
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SMILESCOC1=CC2=NC(NCCCCCC)=NC(NC3CCN(C)CC3)=C2C=C1OC
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Chemical NameN2-Hexyl-6,7-dimethoxy-N4-(1-methylpiperidin-4-yl)quinazoline2,4-diamine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Xiong Y, et al. J Med Chem. 2017 Mar 9;60(5):1876-1891.
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