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MS-023
CAS No. 1831110-54-3
MS-023 ( MS023;MS 023 )
Catalog No. M12819 CAS No. 1831110-54-3
MS-023 is a potent, selective, and cell-active inhibitor of type I PRMTs with IC50s of 30/119/83/4/5 nM for PRMT1/3/4/6/8 respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 42 | In Stock |
|
| 5MG | 72 | In Stock |
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| 10MG | 110 | In Stock |
|
| 25MG | 230 | In Stock |
|
| 50MG | 357 | In Stock |
|
| 100MG | 531 | In Stock |
|
| 500MG | 1152 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameMS-023
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NoteResearch use only, not for human use.
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Brief DescriptionMS-023 is a potent, selective, and cell-active inhibitor of type I PRMTs with IC50s of 30/119/83/4/5 nM for PRMT1/3/4/6/8 respectively.
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DescriptionMS-023 is a potent, selective, and cell-active inhibitor of type I PRMTs with IC50s of 30/119/83/4/5 nM for PRMT1/3/4/6/8 respectively; doesn't inhibit PRMT5/9/7(>10 uM); inhibits H4R3me2a and H3R2me2a levels in MCF7 cells.
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SynonymsMS023;MS 023
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorPRMT1;PRMT3;PRMT4;PRMT6;PRMT8
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Research AreaOther Indications
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Indication——
Chemical Information
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CAS Number1831110-54-3
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Formula Weight287.40
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Molecular FormulaC17H25N3O
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 30 mg/mL
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SMILESCC(C)OC1=CC=C(C=C1)C2=CNC=C2CN(C)CCN
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Chemical Name1,2-Ethanediamine, N1-methyl-N1-[[4-[4-(1-methylethoxy)phenyl]-1H-pyrrol-3-yl]methyl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Eram MS, et al. ACS Chem Biol. 2016 Mar 18;11(3):772-81.
molnova catalog
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