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LEM-14-1189

CAS No.

LEM-14-1189 ( —— )

Catalog No. M17069 CAS No.

LEM-14-1189 is a LEM-14 derivative that differentially inhibits the NSDs.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

LEM-14-1189
Note

Research use only, not for human use.
Brief Description

LEM-14-1189 is a LEM-14 derivative that differentially inhibits the NSDs.
Description

LEM-14-1189 is a LEM-14 derivative that differentially inhibits the NSDs with in vitro IC50 of 418μM (NSD1), IC50 of 111μM (NSD2) and IC50 of 60μM (NSD3).
Synonyms

——
Pathway

Chromatin/Epigenetic
Target

HMTase
Recptor

HMTase
Research Area

——
Indication

——

Chemical Information

CAS Number

--
Formula Weight

682.81
Molecular Formula

C35H34N6O5S2
Purity

>98% (HPLC)
Solubility

——
SMILES

——
Chemical Name

N-(3-(bis((4-oxo-3,4,5,6,7,8-hexahydrobenzo[4,5]thieno[2,3-d]pyrimidin-2-yl)methyl)amino)propyl)-1-oxo-1H-isochromene-3-carboxamide

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Shen Y, et al. Biochem Biophys Res Commun. 2018 Nov 21. pii: S0006-291X(18)32443-4.

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