MRS1186

CAS No. 183721-03-1

MRS1186( MRS-1186 )

Catalog No. M12837 CAS No. 183721-03-1

MRS1186 (MRS-1186) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist with Ki of 7.66 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    MRS1186
  • Note
    Research use only, not for human use.
  • Brief Description
    MRS1186 (MRS-1186) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist with Ki of 7.66 nM.
  • Description
    MRS1186 (MRS-1186) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist with Ki of 7.66 nM.
  • In Vitro
    MRS1186 (compound 2d) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM.
  • In Vivo
    ——
  • Synonyms
    MRS-1186
  • Pathway
    Apoptosis
  • Target
    Adenosine Receptor
  • Recptor
    Adenosine Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    183721-03-1
  • Formula Weight
    341.755
  • Molecular Formula
    C16H12ClN5O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CCC(NC1=NC2=C(C=C(Cl)C=C2)C3=NC(C4=CC=CO4)=NN13)=O
  • Chemical Name
    N-(9-chloro-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)propionamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Tafi A, et al. J Med Chem. 2006 Jul 13;49(14):4085-97.
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