Cart
sales@molnova.com
MRS1186
CAS No. 183721-03-1
MRS1186( MRS-1186 )
Catalog No. M12837 CAS No. 183721-03-1
MRS1186 (MRS-1186) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist with Ki of 7.66 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | Get Quote |
|
| 50MG | 1782 | Get Quote |
|
| 100MG | 2250 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameMRS1186
-
NoteResearch use only, not for human use.
-
Brief DescriptionMRS1186 (MRS-1186) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist with Ki of 7.66 nM.
-
DescriptionMRS1186 (MRS-1186) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist with Ki of 7.66 nM.
-
In VitroMRS1186 (compound 2d) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM.
-
In Vivo——
-
SynonymsMRS-1186
-
PathwayApoptosis
-
TargetAdenosine Receptor
-
RecptorAdenosine Receptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number183721-03-1
-
Formula Weight341.755
-
Molecular FormulaC16H12ClN5O2
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCCC(NC1=NC2=C(C=C(Cl)C=C2)C3=NC(C4=CC=CO4)=NN13)=O
-
Chemical NameN-(9-chloro-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)propionamide
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Tafi A, et al. J Med Chem. 2006 Jul 13;49(14):4085-97.
molnova catalog
related products
-
Neladenoson dalanate
Neladenoson dalanate is a potent, selective, orally acitve partial adenosine A1 receptor (A1AR) agonist (EC50=0.1 nM).
-
Pentoxifylline
A METHYLXANTHINE derivative that inhibits phosphodiesterase and affects blood rheology.
-
Istradefylline
A potent and highly selective A2A receptor antagonist with Ki of 2.2 nM.
