ML179
CAS No. 1883548-87-5
ML179( ML-179 )
Catalog No. M23858 CAS No. 1883548-87-5
ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 110 | In Stock |
|
| 10MG | 177 | In Stock |
|
| 25MG | 368 | In Stock |
|
| 50MG | 536 | In Stock |
|
| 100MG | 779 | In Stock |
|
| 500MG | 1593 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameML179
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NoteResearch use only, not for human use.
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Brief DescriptionML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.
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DescriptionML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.
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In Vitro——
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In Vivo——
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SynonymsML-179
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PathwayOthers
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TargetOther Targets
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Recptorliver receptor homolog-1 (LRH1, NR5A2)
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Research Area——
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Indication——
Chemical Information
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CAS Number1883548-87-5
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Formula Weight424.5
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Molecular FormulaC21H27F3N4O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 12.5 mg/mL (29.59 mM)
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SMILESC1CCC(CC1)N2C(=O)CC(NC2=O)N3CCN(CC3)C4=CC=CC(=C4)C(F)(F)F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Busby S , Nuhant P , Ca Meron M , et al. Discovery of Inverse Agonists for the Liver Receptor Homologue-1 (LRH1; NR5A2)[M]. PubMed, 2010.
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