ML179

CAS No. 1883548-87-5

ML179( ML-179 )

Catalog No. M23858 CAS No. 1883548-87-5

ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 110 In Stock
10MG 177 In Stock
25MG 368 In Stock
50MG 536 In Stock
100MG 779 In Stock
500MG 1593 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    ML179
  • Note
    Research use only, not for human use.
  • Brief Description
    ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.
  • Description
    ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ML-179
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    liver receptor homolog-1 (LRH1, NR5A2)
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1883548-87-5
  • Formula Weight
    424.5
  • Molecular Formula
    C21H27F3N4O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 12.5 mg/mL (29.59 mM)
  • SMILES
    C1CCC(CC1)N2C(=O)CC(NC2=O)N3CCN(CC3)C4=CC=CC(=C4)C(F)(F)F
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Busby S , Nuhant P , Ca Meron M , et al. Discovery of Inverse Agonists for the Liver Receptor Homologue-1 (LRH1; NR5A2)[M]. PubMed, 2010.
molnova catalog
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