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MEDICA16
CAS No. 87272-20-6
MEDICA16( MEDICA 16 )
Catalog No. M27653 CAS No. 87272-20-6
MEDICA16 is a selective agonist for GPR40 as well as a partial agonist for GPR120.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 87 | Get Quote |
|
| 10MG | 132 | Get Quote |
|
| 25MG | 282 | Get Quote |
|
| 50MG | 484 | Get Quote |
|
| 100MG | 700 | Get Quote |
|
| 500MG | 1458 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameMEDICA16
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NoteResearch use only, not for human use.
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Brief DescriptionMEDICA16 is a selective agonist for GPR40 as well as a partial agonist for GPR120.
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DescriptionMEDICA16 is a selective agonist for GPR40 as well as a partial agonist for GPR120. MEDICA16, an ATP-citrate lyase inhibitor, significantly reduces intracellular TG content in gastrocnemius muscle with an increase in insulin sensitivity.
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In Vitro——
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In Vivo——
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SynonymsMEDICA 16
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PathwayCell Cycle/DNA Damage
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TargetGPR
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RecptorPHD3|HIF-2α|VEGFR1
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Research Area——
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Indication——
Chemical Information
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CAS Number87272-20-6
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Formula Weight342.52
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Molecular FormulaC20H38O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (291.96 mM)
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SMILESCC(C)(CCCCCCCCCCC(C)(C)CC(O)=O)CC(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Roda JM, et al. Stabilization of HIF-2α induces sVEGFR-1 production from tumor-associated macrophages and decreases tumor growth in a murine melanoma model. J Immunol. 2012 Sep 15;189(6):3168-77.
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