Cart
sales@molnova.com
Home - Products - Cell Cycle/DNA Damage - PARP - ARTD10/PARP10-IN-1

ARTD10/PARP10-IN-1

CAS No. 1708103-76-7

ARTD10/PARP10-IN-1( —— )

Catalog No. M36466 CAS No. 1708103-76-7

ARTD10/PARP10-IN-1 is a potent PARP inhibitor of the mono-ADP ribosyltransferases ARTD7/PARP15, ARTD8/PARP14, ARTD10/PARP10 and poly ADP-ribose polymerase-1 (ARTD1/PARP1), with potential anticancer and antitumour activity for the study of prostate and breast cancers.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 645 In Stock
10MG 772 In Stock
25MG 969 In Stock
50MG 1283 In Stock
100MG 1628 In Stock
200MG 2167 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    ARTD10/PARP10-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    ARTD10/PARP10-IN-1 is a potent PARP inhibitor of the mono-ADP ribosyltransferases ARTD7/PARP15, ARTD8/PARP14, ARTD10/PARP10 and poly ADP-ribose polymerase-1 (ARTD1/PARP1), with potential anticancer and antitumour activity for the study of prostate and breast cancers.
  • Description
    ARTD10/PARP10-IN-1 (compound 23) is a potent and non-selective PARP inhibitor, targeting to mono-ADP-ribosyltransferases ARTD7/PARP15, ARTD8/PARP14, ARTD10/PARP10 and poly(ADP-ribose) polymerase-1 (ARTD1/PARP1) with IC50s of 1.7 μM, 1.6 μM, 0.8 μM, and 4.4 μM, respectively.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    PARP
  • Recptor
    PARP
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1708103-76-7
  • Formula Weight
    248.23
  • Molecular Formula
    C12H12N2O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    N(C(/C=C\C(OC)=O)=O)C1=CC(C(N)=O)=CC=C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Ekblad T, et al. Towards small molecule inhibitors of mono-ADP-ribosyltransferases. Eur J Med Chem. 2015 May 5;95:546-51.?
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • NVP-BVU972

    NVP-BVU972 is a selective and potent Met inhibitor with IC50 of 14 nM.

  • 2-CHLORO-5-CYANOPYRA...

    2-CHLORO-5-CYANOPYRAZINE is an active biochemical.

  • Venadaparib

    Venadaparib (IDX-1197) is a potent, selective and orally active PARP inhibitor with IC50s of 1.4 nM and 1.0 nM for PARP1 and PARP2, respectively.

Sign In Join Free