CTX-0124143

CAS No. 423731-64-0

CTX-0124143( —— )

Catalog No. M36385 CAS No. 423731-64-0

CTX-0124143 is a histone acetyltransferase inhibitor with an IC50 value of 1.0 μM for KAT6A.CTX-0124143 can be used to study cellular senescence.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 70 In Stock
10MG 113 In Stock
25MG 210 In Stock
50MG 319 In Stock
100MG 421 In Stock
200MG 568 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    CTX-0124143
  • Note
    Research use only, not for human use.
  • Brief Description
    CTX-0124143 is a histone acetyltransferase inhibitor with an IC50 value of 1.0 μM for KAT6A.CTX-0124143 can be used to study cellular senescence.
  • Description
    CTX-0124143 is a KAT6A inhibitor with a sulfonyl hydrazine skeleton.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Histone Acetyltransferase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    423731-64-0
  • Formula Weight
    344.36
  • Molecular Formula
    C17H13FN2O3S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 125 mg/mL (362.99 mM; Ultrasonic )
  • SMILES
    FC1=C(C=CC=C1)C(=O)NNS(=O)(=O)C1=CC2=CC=CC=C2C=C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Duan Y, et al. Discovery of N-(2-oxoethyl) sulfanilamide-derived inhibitors of KAT6A (MOZ) against leukemia by an isostere strategy. Eur J Med Chem. 2023 Nov 15;260:115770.?
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