CTX-0124143
CAS No. 423731-64-0
CTX-0124143( —— )
Catalog No. M36385 CAS No. 423731-64-0
CTX-0124143 is a histone acetyltransferase inhibitor with an IC50 value of 1.0 μM for KAT6A.CTX-0124143 can be used to study cellular senescence.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 70 | In Stock |
|
| 10MG | 113 | In Stock |
|
| 25MG | 210 | In Stock |
|
| 50MG | 319 | In Stock |
|
| 100MG | 421 | In Stock |
|
| 200MG | 568 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameCTX-0124143
-
NoteResearch use only, not for human use.
-
Brief DescriptionCTX-0124143 is a histone acetyltransferase inhibitor with an IC50 value of 1.0 μM for KAT6A.CTX-0124143 can be used to study cellular senescence.
-
DescriptionCTX-0124143 is a KAT6A inhibitor with a sulfonyl hydrazine skeleton.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayOthers
-
TargetOther Targets
-
RecptorHistone Acetyltransferase
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number423731-64-0
-
Formula Weight344.36
-
Molecular FormulaC17H13FN2O3S
-
Purity>98% (HPLC)
-
SolubilityIn Vitro:?DMSO : 125 mg/mL (362.99 mM; Ultrasonic )
-
SMILESFC1=C(C=CC=C1)C(=O)NNS(=O)(=O)C1=CC2=CC=CC=C2C=C1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Duan Y, et al. Discovery of N-(2-oxoethyl) sulfanilamide-derived inhibitors of KAT6A (MOZ) against leukemia by an isostere strategy. Eur J Med Chem. 2023 Nov 15;260:115770.?
molnova catalog
related products
-
InsB 9-23
InsB (9-23) is an insulin B-chain peptide that binds to a class II histocompatibility complex (MHC) allele called I-Ag7.
-
guan-fu base H
Guanfu base H (Atisinium chloride) is a diterpenoid alkaloid isolated from Aconitum coreanum and has antiplasmodial activity against the malarial Plasmodium falciparum strains TM4/8.2 (wild type) and K1CB1 with IC50 values of 4 μM and 3.6 μM, respectively.
-
SMA-12b
SMA-12b is an analog of the immunomodulatory parasite product ES-62 that has immunomodulatory activity, can modify the expression of many inflammatory response genes.
Cart
sales@molnova.com