UNC?1021

CAS No. 1322591-19-4

UNC?1021( —— )

Catalog No. M35814 CAS No. 1322591-19-4

UNC 1021 is a selective L3MBTL3 inhibitor (IC50 = 0.048 μM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 36 In Stock
10MG 55 In Stock
25MG 107 In Stock
50MG 166 In Stock
100MG 267 In Stock
200MG 369 In Stock
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Biological Information

  • Product Name
    UNC?1021
  • Note
    Research use only, not for human use.
  • Brief Description
    UNC 1021 is a selective L3MBTL3 inhibitor (IC50 = 0.048 μM).
  • Description
    UNC1021 is a selective L3MBTL3 inhibitor with an IC50 of 0.048 μM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Chromatin/Epigenetic
  • Target
    Epigenetic Reader Domain
  • Recptor
    Epigenetic Reader Domain
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1322591-19-4
  • Formula Weight
    438.61
  • Molecular Formula
    C26H38N4O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : ≥ 9.09 mg/mL (20.72 mM )
  • SMILES
    O=C(N1CCC(CC1)N1CCCC1)c1ccc(cc1)C(=O)N1CCC(CC1)N1CCCC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. James LI, et al. Small-molecule ligands of methyl-lysine binding proteins: optimization of selectivity for L3MBTL3. J Med Chem. 2013 Sep 26;56(18):7358-71.?
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