FGFR2-IN-1

CAS No. 2677709-76-9

FGFR2-IN-1( —— )

Catalog No. M35540 CAS No. 2677709-76-9

FGFR2-IN-1 is an FGFR inhibitor that inhibits FGFR1, FGFR2, and FGFR3 with IC50s of 460, 140, and 2200 nM, respectively.FGFR2-IN-1 can be used for the study of cancers associated with FGFR2.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 85 Get Quote
5MG 128 Get Quote
10MG 202 Get Quote
25MG 330 Get Quote
50MG 490 Get Quote
100MG 683 Get Quote
500MG 1377 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    FGFR2-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    FGFR2-IN-1 is an FGFR inhibitor that inhibits FGFR1, FGFR2, and FGFR3 with IC50s of 460, 140, and 2200 nM, respectively.FGFR2-IN-1 can be used for the study of cancers associated with FGFR2.
  • Description
    FGFR2-IN-1 is a selective FGFR2 inhibitor with an IC50 of 140 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    FGFR
  • Recptor
    FGFR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2677709-76-9
  • Formula Weight
    357.41
  • Molecular Formula
    C22H19N3O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(NC1=NNC=2C=C(C=CC12)C=3C=CC=C(OCC)C3)C=4C=CC=CC4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Turner LD, et al. From Fragment to Lead: De Novo Design and Development toward a Selective FGFR2 Inhibitor. J. Med. Chem. 2021 Nov 15.
molnova catalog
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