FGFR4-IN-1

CAS No. 1708971-72-5

FGFR4-IN-1( —— )

Catalog No. M23769 CAS No. 1708971-72-5

FGFR4-IN-1 is a potent FGFR4 inhibitor (IC50: 0.7 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 92 In Stock
5MG 92 In Stock
10MG 148 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    FGFR4-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    FGFR4-IN-1 is a potent FGFR4 inhibitor (IC50: 0.7 nM).
  • Description
    FGFR4-IN-1 is a potent FGFR4 inhibitor (IC50: 0.7 nM).
  • In Vitro
    FGFR4-IN-1 significantly inhibits the proliferation of HuH-7 hepatocellular carcinoma cells with IC50 of 7.8 nM.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    FGFR
  • Recptor
    FGFR4
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1708971-72-5
  • Formula Weight
    493.52
  • Molecular Formula
    C24H27N7O5
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:6 mg/mL (12.16 mM; Need warming)
  • SMILES
    COCCNc1cc(NC(N2c3nc(C=O)c(CN(CCOC4)C4=O)cc3CCC2)=O)ncc1C#N
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ring-fused bicyclic pyridyl derivatives as fgfr4 inhibitors. WO 2015059668 A1
molnova catalog
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